Synthesis of a 10 000 Member 1,5-Benzodiazepine-2-one Library by the Directed Sorting Method
- 13 July 2000
- journal article
- research article
- Published by American Chemical Society (ACS) in Journal of Combinatorial Chemistry
- Vol. 2 (5) , 513-521
- https://doi.org/10.1021/cc000025u
Abstract
No abstract availableKeywords
This publication has 10 references indexed in Scilit:
- Solid-phase synthesis of 1,5-benzodiazepin-2-onesTetrahedron Letters, 1998
- Class III Antiarrhythmic Activity in Vivo by Selective Blockade of the Slowly Activating Cardiac Delayed Rectifier Potassium Current IKs by (R)-2-(2,4- Trifluoromethyl)-N-[2-oxo-5-phenyl- 1-(2,2,2-trifluoroethyl)-2,3-dihydro- 1H-benzo[e][1,4]diazepin-3-yl]acetamideJournal of Medicinal Chemistry, 1997
- Solid-Phase Synthesis of 1,4-Benzodiazepine-2,5-diones. Library Preparation and Demonstration of Synthesis GeneralityThe Journal of Organic Chemistry, 1997
- Novel 1,5‐Benzodiazepines as CCK‐B Ligands. Effect of Aryl‐Carbamic Substituents at the C‐3 Position Together with Halogen Substitution on the Benzo‐Fused RingArchiv der Pharmazie, 1997
- An expedient and high-yielding method for the solid-phase synthesis of diverse 1,4-benzodiazepine-2,5-dionesThe Journal of Organic Chemistry, 1995
- Solid-Phase Synthesis of Structurally Diverse 1,4-Benzodiazepine Derivatives Using the Stille Coupling ReactionJournal of the American Chemical Society, 1995
- A general and expedient method for the solid-phase synthesis of 1,4-benzodiazepine derivativesJournal of the American Chemical Society, 1992
- Methods for drug discovery: development of potent, selective, orally effective cholecystokinin antagonistsJournal of Medicinal Chemistry, 1988
- Diazepam-Binding Inhibitor: A Neuropeptide Located in Selected Neuronal Populations of Rat BrainScience, 1985
- Relationship of β-adrenoreceptor density to fitness in athletesNature, 1982