5-HT2A, 5-HT2B and 5-HT2C receptor ligands
- 1 January 1997
- book chapter
- Published by Elsevier
Abstract
No abstract availableThis publication has 52 references indexed in Scilit:
- 5-Methyl-1-(3-pyridylcarbamoyl)-1,2,3,5-tetrahydropyrrolo[2,3-f]indole: A Novel 5-HT2C/5-HT2B Receptor Antagonist with Improved Affinity, Selectivity, and Oral ActivityJournal of Medicinal Chemistry, 1995
- The Third Intracellular Loop of the 5‐Hydroxytryptamine2A Receptor Determines Effector Coupling SpecificityJournal of Neurochemistry, 1995
- Ketanserin Analogs: The Effect of Structural Modification on 5-HT2 Serotonin Receptor BindingJournal of Medicinal Chemistry, 1995
- 3-[[(Aryloxy)alkyl]piperidinyl]-1,2-Benzisoxazoles as D2/5-HT2 Antagonists with Potential Atypical Antipsychotic Activity: Antipsychotic Profile of Iloperidone (HP 873)Journal of Medicinal Chemistry, 1995
- Stereospecific and selective 5-HT2 antagonism in a series of 5-substituted trans-1-piperazino-3-phenylindansJournal of Medicinal Chemistry, 1993
- 1-(2-Aminoethyl)-3-methyl-8,9-dihydropyrano[3,2-e]indole: a rotationally restricted phenolic analog of the neurotransmitter serotonin and agonist selective for serotonin (5-HT2-type) receptorsJournal of Medicinal Chemistry, 1992
- Site‐directed mutagenesis of a single residue changes the binding properties of the serotonin 5‐HT2 receptor from a human to a rat pharmacologyFEBS Letters, 1992
- Naphthosultam derivatives: a new class of potent and selective 5-HT2 antagonistsJournal of Medicinal Chemistry, 1991
- The concept of selectivity in 5-HT receptor researchEuropean Journal of Pharmacology: Molecular Pharmacology, 1990
- (8.beta.)-Ergoline-8-carboxylic acid cycloalkyl esters as serotonin antagonists: structure-activity studyJournal of Medicinal Chemistry, 1988