Design and synthesis of novel 2,3-dihydro-1H-isoindoles with high affinity and selectivity for the dopamine D3 receptor
- 8 March 2001
- journal article
- research article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 11 (5) , 685-688
- https://doi.org/10.1016/s0960-894x(01)00037-3
Abstract
No abstract availableKeywords
This publication has 9 references indexed in Scilit:
- Design and Synthesis of trans-N-[4-[2-(6-Cyano-1,2,3,4-tetrahydroisoquinolin-2- yl)ethyl]cyclohexyl]-4-quinolinecarboxamide (SB-277011): A Potent and Selective Dopamine D3 Receptor Antagonist with High Oral Bioavailability and CNS Penetration in the RatJournal of Medicinal Chemistry, 2000
- Selective inhibition of cocaine-seeking behaviour by a partial dopamine D3 receptor agonistNature, 1999
- Novel 1,2,3,4-tetrahydroisoquinolines with high affinity and selectivity for the dopamine D3 receptorBioorganic & Medicinal Chemistry Letters, 1999
- The D 3 dopamine receptor in cellular and organismal functionPsychopharmacology, 1998
- A novel series of 2-aminotetralins with high affinity and selectivity for the dopamine D3 receptorBioorganic & Medicinal Chemistry Letters, 1997
- Linking the Family of D2 Receptors to Neuronal Circuits in Human Brain: Insights into SchizophreniaNeuropsychopharmacology, 1997
- Design and Synthesis of 2-Naphthoate Esters as Selective Dopamine D4AntagonistsJournal of Medicinal Chemistry, 1996
- Dopamine D3 Receptor: Basic and Clinical AspectsClinical Neuropharmacology, 1993
- Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neurolepticsNature, 1990