The Use of Lewis Acid in the Reaction of Zinc Salts of Indoles and Acyl Chloride
- 1 June 1997
- journal article
- research article
- Published by Taylor & Francis in Synthetic Communications
- Vol. 27 (12) , 2125-2132
- https://doi.org/10.1080/00397919708006820
Abstract
3-Acylindoles have been prepared in 62 – 92% isolated yield from the corresponding indoles and acyl chlorides in the presence of AlCl3.Keywords
This publication has 10 references indexed in Scilit:
- N-(Acyloxyalkyl)pyridinium Salts as Soluble Prodrugs of a Potent Platelet Activating Factor AntagonistJournal of Medicinal Chemistry, 1994
- 3-(2-(3-Pyridinyl)thiazolidin-4-oyl)indoles, a Novel Series of Platelet Activating Factor AntagonistsJournal of Medicinal Chemistry, 1994
- Formation of 6-acylindoles from 1-acylindolesTetrahedron Letters, 1994
- Synthesis of 6- and 7-ArylindolesviaPalladium-Catalyzed Cross-Coupling of 6- and 7-Bromoindole with Arylboronic AcidsSynlett, 1994
- Thiomethylation of indole and haloindole zinc saltsTetrahedron Letters, 1993
- Acylation of the zinc salt of indoleTetrahedron, 1990
- Yuehchukene analogsThe Journal of Organic Chemistry, 1988
- Intramolecular, ring closure of α,β-unsaturated 3-acylindolesTetrahedron Letters, 1987
- A convenient synthesis of 3-acylindoles via Friedel Crafts acylation of 1-(phenylsulfonyl)indole. A new route to pyridocarbazole-5,11-quinones and ellipticineThe Journal of Organic Chemistry, 1985
- Notes- Novel Synthesis of Heterocyclic KetonesThe Journal of Organic Chemistry, 1960