ASYMMETRIC SYNTHESIS OF 1-AMINOALKYLPHOSPHONIC ACIDS
- 1 January 1993
- journal article
- research article
- Published by Taylor & Francis in Phosphorus, Sulfur, and Silicon and the Related Elements
- Vol. 81 (1-4) , 83-87
- https://doi.org/10.1080/10426509308034376
Abstract
Asymmetric synthesis of Phe and Tyr phosphonic analogous has been achieved by diastereoselective alkylation of chiral 1,2,3-oxazaphospholanes, the latter being readily obtained from (-) ephedrine and chloromethylphosphonic dichloride.Keywords
This publication has 8 references indexed in Scilit:
- Asymmetric electrophilic amination of chiral phosphorus-stabilized anionsTetrahedron, 1992
- Studies toward a model for predicting the diastereoselectivity in the electrophilic amination of chiral 1,3,2-oxazaphospholanesTetrahedron, 1992
- A versatile asymmetric synthesis of α-amino α-alkyl-phosphonic acids of high enantiomeric purityTetrahedron Letters, 1990
- Phosphoranaloge von Aminosäuren III1. Synthese optisch aktiver 1-Aminoalkylphosphonsäuren der (S)- und (R)-Reihe mit Hilfe von (-)-Ephedrin als AuxiliarSynthesis, 1990
- OPTICALLY ACTIVE 1-AMINOALKYLPHOSPHONIC ACIDSPhosphorus, Sulfur, and Silicon and the Related Elements, 1987
- 1,3,2-Oxazaphospholidines from (–)-ephedrine. Intermediates for the stereospecific synthesis of optically active dialkyl alkylphosphonothioates and -selenoates, trialkyl phosphoro-thioates and -selenoates, dialkyl methylphosphonates, and trialkyl phosphatesJournal of the Chemical Society, Perkin Transactions 1, 1977
- Preparation, stereochemistry and some reactions of 1,3,2-oxazaphospholanesTetrahedron Letters, 1974
- Peptides Containing Aminophosphonic Acids. II. The Synthesis of Tripeptide AnalogsBulletin of the Chemical Society of Japan, 1972