A Facile Synthesis of 2-N(Methyl Amino) Benzothiazoles
- 1 May 1997
- journal article
- research article
- Published by Taylor & Francis in Synthetic Communications
- Vol. 27 (9) , 1487-1493
- https://doi.org/10.1080/00397919708006084
Abstract
Reaction of aromatic primary amines with methylisothiocyanate (MITC) yielded N-methyl-N1-(benzelene-1-yl)thioureas which underwent oxidative cyclization in the presence of bromine in acetic acid, at room temperature, affording the title compounds.Keywords
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