Studies on Local Anesthetics. XIX. Local Anesthetic Activity of N-(Dialkylaminoalkyl)benzamides. Physicochemical Measurements on N-(Dialkylaminoalkyl)benzamides and Benzoic Acid.

Abstract
Local anesthetic properties and LD50 values were evaluated for 26 N-(dialkylaminoalkyl)benzamides. Ionization constants were determined for 26 N-(dialkylaminoalkyl)benzamides, for benzoic acid and all mono, di-, and trimethylbenzoic acids. Ultraviolet spectra were measured on 15 N-(dialkylaminoalkyl)benzamides, 5 dimethyl-, and all trimethylbenzoic acids. The oscillator strength of these compounds for the absorption band at 220-240 m[mu] was determined and a correlation between these values and the ionization constants was found. Infrared spectra were recorded for the two racemates of N-(2-diethylamino-l,2-dimethylethyl)-2-methylbenzamide.

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