Asymmetric synthesis of building-blocks for peptides and peptidomimetics by means of the β-lactam synthon method
- 1 January 1997
- journal article
- Published by Royal Society of Chemistry (RSC) in Chemical Society Reviews
- Vol. 26 (5) , 377-386
- https://doi.org/10.1039/cs9972600377
Abstract
Recent advances in the syntheses of enantiopure synthetic building blocks useful for non-protein amino acids, dipeptides, oligopeptides using solid state peptide synthesis, isoserines (norstatines), dipeptide isosteres [hydroxy(keto)ethylene, hydroxyethylamine, hydroxyethylene and dihydroxyethylene isosteres], taxoids, polyamines, poly(amino alcohol)s and poly(amino ether)s, and other biologically active compounds through applications of the β-lactam Synthon method is reviewed.Keywords
This publication has 26 references indexed in Scilit:
- Application of (+)-(1S,2S)-2-amino-1-phenylpropan-1,3-diol in the formal total synthesis of carbapenems, novel 4-cyano-β-lactams and β-hydroxy aspartatesTetrahedron, 1996
- 1(2,6-dichlorophenyl)ethylamine: a new and efficient chiral auxiliary for the Staudinger β-lactam synthesisTetrahedron Letters, 1995
- Recent Advances in the .beta.-Lactam Synthon MethodAccounts of Chemical Research, 1995
- An investigation of (R)-(+)-1-(1-naphthyl)ethylimines and (R)-(+)-1-(phenyl)ethylimines as chiral templates in the staudinger reactionTetrahedron Letters, 1994
- Stereoregulated synthesis of β-lactams from schiff bases derived from threonine estersTetrahedron, 1992
- Enantioselective synthesis of a versatile 2-isocephem synthonTetrahedron, 1990
- Remarkable effects of lone pair-lone pair interactions on the extremely stereoselective [2 + 2] cycloaddition of azidoketene to chiral 3-imino-.beta.-lactamsJournal of the American Chemical Society, 1987
- Chiral control of the Staudinger reactionPublished by Walter de Gruyter GmbH ,1987
- The asymmetric synthesis of β-lactam antibiotics - I. application of chiral oxazolidones in the staudinger reaction.Tetrahedron Letters, 1985
- Synthetic Studies on Optically Active b-Lactams. Asymmetric Synthesis of b-Lactams by the Cyclocondensation Utilizing Chiral Heterocyclic Compounds Derived from L-(+)-Tartaric Acid and (S)-Glutamic AcidHETEROCYCLES, 1984