Alternatives to Vinyl Triflates for Cross-Coupling with Arylboronic Acids

Abstract
Vinyl phosphates, mesylates, and tosylates derived from 1,3-dicarbonyl compounds are coupled with phenylboronic acid using nickel or palladium catalysts. An application to the area of 2-aryl carbapenem antibiotics is demonstrated. Alternative conditions for the nickel-catalyzed coupling of aryl mesylates are also reported.

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