Preparation of α-Halo-α,β-Unsaturated Bicyclic Lactams and Their Use in Palladium-Catalyzed Cross Coupling Reactions

1 January 1993

journal article
letter
Published by Georg Thieme Verlag KG in Synlett

Vol. 1993 (08) , 573-574
https://doi.org/10.1055/s-1993-22533

Abstract

Efficient syntheses of α-halo-α,β-unsaturated lactams from the corresponding saturated and unsaturated lactams are described. These substrates undergo palladium-catalyzed Stille and Suzuki couplings, furnishing α-substituted-α,β-unsaturated lactams in good yields.

Keywords

Α HALO
Β UNSATURATED
STILLE
UNDERGO
GOOD

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