Chiral synthesis of statine
- 31 December 1985
- journal article
- Published by Elsevier in Tetrahedron Letters
- Vol. 26 (25) , 2973-2976
- https://doi.org/10.1016/s0040-4039(00)98595-2
Abstract
No abstract availableKeywords
This publication has 16 references indexed in Scilit:
- Pepstatin-derived inhibitors of aspartic proteinases. A close look at an apparent transition-state analog inhibitorJournal of Medicinal Chemistry, 1985
- Novel renin inhibitors containing the amino acid statineNature, 1983
- An Efficient Synthesis of Optically Active α-(t-Butoxycarbonylamino)-aldehydes from α-Amino AcidsSynthesis, 1983
- A synthesis of statine utilizing an oxidative route to chiral .alpha.-amino aldehydesThe Journal of Organic Chemistry, 1982
- Stereoselective aldol condensations via boron enolatesJournal of the American Chemical Society, 1981
- Enantioselective aldol condensations. 2. Erythro-selective chiral aldol condensations via boron enolatesJournal of the American Chemical Society, 1981
- Synthesis of all the stereoisomers of statine (4-amino-3-hydroxy-6-methylheptanoic acid). Inhibition of pepsin activity by N-carbobenzoxy-L-valyl-L-valyl-statine derived from the four stereoisomersJournal of Medicinal Chemistry, 1979
- Synthesis of (3S,4S)-4-amino-3-hydroxy-6-methylheptanoic acid derivatives. Analysis of diastereomeric purityThe Journal of Organic Chemistry, 1978
- Synthesis of 4-amino-3-hydroxy-6-methylheptanoic acid by a modified Reformatsky reactionThe Journal of Organic Chemistry, 1978
- Synthesis of (3S, 4S)- and (3S, 4R)-4-Amino-3-hydroxy-6-methylheptanoic Acid, and Their N-(Acetyl-l-valyl-l-valyl) DerivativesBulletin of the Chemical Society of Japan, 1975