Synthesis and radiolabeling of N-[4-[4-(2-[11C]methoxyphenyl)piperazin-1-yl]butyl]benzo[b]thiophene-2-carboxamide — a potential radiotracer for D3 receptor imaging with PET
- 1 August 2006
- journal article
- Published by Elsevier in Nuclear Medicine and Biology
- Vol. 33 (6) , 785-795
- https://doi.org/10.1016/j.nucmedbio.2006.05.007
Abstract
No abstract availableKeywords
This publication has 43 references indexed in Scilit:
- Dopamine D3 receptor antagonists as therapeutic agentsDrug Discovery Today, 2005
- The role of central dopamine D3 receptors in drug addiction: a review of pharmacological evidenceBrain Research Reviews, 2005
- Novel Heterocyclic Trans Olefin Analogues of N-{4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl}arylcarboxamides as Selective Probes with High Affinity for the Dopamine D3 ReceptorJournal of Medicinal Chemistry, 2005
- Protection against Cocaine Toxicity in Mice by the Dopamine D3/D2 Agonist R-(+)-trans-3,4 a,10 b-Tetrahydro-4-propyl-2 H,5 H-[1]benzopyrano[4,3-b]-1,4-oxazin-9-ol [(+)-PD 128,907]The Journal of Pharmacology and Experimental Therapeutics, 2004
- Conformationally-flexible benzamide analogues as dopamine D3 and σ2 receptor ligandsBioorganic & Medicinal Chemistry Letters, 2003
- Synthesis and Pharmacological Evaluation of Potent and Highly Selective D3 Receptor Ligands: Inhibition of Cocaine-Seeking Behavior and the Role of Dopamine D3/D2 ReceptorsJournal of Medicinal Chemistry, 2003
- Disruption of nicotine conditioning by dopamine D3 receptor ligandsMolecular Psychiatry, 2003
- Dopamine D3 Receptor Ligands with Antagonist PropertiesChemBioChem, 2002
- The dopamine D3 receptor and drug addictionNeurotoxicity Research, 2001
- Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neurolepticsNature, 1990