Synthesis of new thiazinoindole derivatives and their evaluation as inhibitors of human leukocyte elastase and other related serine proteases
- 1 October 1994
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 4 (20) , 2399-2404
- https://doi.org/10.1016/s0960-894x(01)80398-x
Abstract
No abstract availableKeywords
This publication has 14 references indexed in Scilit:
- Specificity, stability, and potency of monocyclic .beta.-lactam inhibitors of human leukocyte elastaseBiochemistry, 1992
- Synthesis of novel 1,3-oxazino[6,5-b]indole-2,4-(3H,9H)-dione and 2H-1,3,5-oxadiazino[3,2-a]indole-2,4-(3H)-dione from oxindolesJournal of Heterocyclic Chemistry, 1992
- Design and synthesis of 4H-3,1-benzoxazin-4-ones as potent alternate substrate inhibitors of human leukocyte elastaseJournal of Medicinal Chemistry, 1990
- Granulocyte Neutral Proteases and Pseudomonas Elastase as Possible Causes of Airway Damage in Patients with Cystic FibrosisThe Journal of Infectious Diseases, 1984
- Interactions of Granulocyte Proteases with Inhibitors in Rheumatoid ArthritisPublished by Springer Nature ,1984
- Low Molecular Mass Bronchial Proteinase Inhibitor and α1-Proteinase Inhibitor in Sputum and Bronchoalveolar LavageHoppe-Seyler´s Zeitschrift Für Physiologische Chemie, 1984
- Elastase and alpha 1-proteinase inhibitor activity in tracheal aspirates during respiratory distress syndrome. Role of inflammation in the pathogenesis of bronchopulmonary dysplasia.Journal of Clinical Investigation, 1983
- New class of serine protease inactivators based on isatoic anhydrideJournal of the American Chemical Society, 1982
- Acylanthranils. 3. The influence of ring substituents on reactivity and selectivity in the reaction of acylanthranils with aminesThe Journal of Organic Chemistry, 1977
- Structure of crystalline α-chymotrypsinJournal of Molecular Biology, 1970