A novel bifunctional maleimido CHX-A″ chelator for conjugation to thiol-containing biomolecules
- 15 April 2008
- journal article
- research article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 18 (8) , 2679-2683
- https://doi.org/10.1016/j.bmcl.2008.03.022
Abstract
No abstract availableKeywords
This publication has 19 references indexed in Scilit:
- Design, Synthesis, and Characterization of a Dual Modality Positron Emission Tomography and Fluorescence Imaging Agent for Monoclonal Antibody Tumor-Targeted ImagingJournal of Medicinal Chemistry, 2007
- Potentiation of High-LET Radiation by Gemcitabine: Targeting HER2 with Trastuzumab to Treat Disseminated Peritoneal DiseaseClinical Cancer Research, 2007
- Validation of a Novel CHX-A‘ ‘ Derivative Suitable for Peptide Conjugation: Small Animal PET/CT Imaging Using Yttrium-86-CHX-A‘ ‘-OctreotideJournal of Medicinal Chemistry, 2006
- Arming antibodies: prospects and challenges for immunoconjugatesNature Biotechnology, 2005
- Targeting of HER2 Antigen for the Treatment of Disseminated Peritoneal DiseaseClinical Cancer Research, 2004
- Maleimidocysteineamido-DOTA Derivatives: New Reagents for Radiometal Chelate Conjugation to Antibody Sulfhydryl Groups Undergo pH-Dependent Cleavage ReactionsBioconjugate Chemistry, 1998
- Stereochemical influence on the stability of radio-metal complexes in vivo. Synthesis and evaluation of the four stereoisomers of 2-(p-nitrobenzyl)-trans-CyDTPABioorganic & Medicinal Chemistry, 1997
- Maleimido Derivatives of Diethylenetriaminepentaacetic Acid and Triethylenetetraaminehexaacetic Acid: Their Synthesis and Potential for Specific Conjugation with BiomoleculesBioconjugate Chemistry, 1996
- Spectrophotometric method for the determination of a bifunctional DTPA ligand in DTPA-monoclonal antibody conjugatesBioconjugate Chemistry, 1992
- Addition of sulfhydryl groups of Escherichia coli ribosomes by protein modification with 2-iminothiolane (methyl 4-mercaptobutyrimidate)Biochemistry, 1978