A chemical method for the preparation of novel 1,5-benzodiazepines acting as CCK-B antagonists in high enantiomeric purity
- 1 May 1997
- journal article
- Published by Elsevier in Tetrahedron
- Vol. 53 (21) , 7347-7364
- https://doi.org/10.1016/s0040-4020(97)00418-3
Abstract
No abstract availableKeywords
This publication has 10 references indexed in Scilit:
- Synthesis and evaluation of novel 1,5-Benzodiazepines as potent and selective CCK-B ligands. Effect of the substitution of the N-5 phenyl with alkyl groupsBioorganic & Medicinal Chemistry Letters, 1996
- 1,5-Benzodiazepines as CCK-B antagonists. Effect of halogen substitution at the benzo-fused ring on potency and selectivityBioorganic & Medicinal Chemistry Letters, 1995
- A new method for the resolution of amines and its application to 3-amino-1,5-benzodiazepinesTetrahedron: Asymmetry, 1995
- Carbohydrates as Chiral Auxiliaries in Stereoselective Synthesis. New Synthetic Methods (90)Angewandte Chemie International Edition in English, 1993
- Optically active tetrahydro-.alpha.-phenyl-6,7-dimethoxyisoquinoline-1-methanols from (1-phenylethyl)ureas. Absolute configuration of (-)- and (+)-isomers of the erythro seriesThe Journal of Organic Chemistry, 1989
- A new amine resolution method and its application to 3-aminobenzodiazepinesTetrahedron Letters, 1987
- Synthesis and resolution of 3-amino-1,3-dihydro-5-phenyl-2H-1,4-benzodiazepin-2-onesThe Journal of Organic Chemistry, 1987
- Total synthesis of (.+-.)-solavetivone and aglycone A3. Regio- and stereo-selective Birch reduction of 6,10-dimethyl-2-hydroxy-spiro[4.5]deca-6,9-dien-8-one.CHEMICAL & PHARMACEUTICAL BULLETIN, 1987
- THE TEMPERATURE DEPENDENCE OF HYDROGENOLYTIC ASYMMETRIC TRANSAMINATION BETWEEN ESTERS OF OPTICALLY ACTIVE PHENYLGLYCINE AND PYRUVIC ACIDChemistry Letters, 1978
- The absolute configurations of some .alpha.-thio ethers derived from mandelic acidThe Journal of Organic Chemistry, 1967