Copper(I) Oxide Catalyzed N-Arylation of Azoles and Amines with Arylboronic Acid at Room Temperature under Base-Free Conditions
- 18 February 2008
- journal article
- research article
- Published by Georg Thieme Verlag KG in Synthesis
- Vol. 2008 (5) , 795-799
- https://doi.org/10.1055/s-2008-1032184
Abstract
N-Arylation of azoles and amines with arylboronic acids was efficiently carried out with heterogeneous copper(I) oxide in methanol at room temperature under base-free conditions. The products N-arylazoles and N-arylamines were isolated in good to excellent yields. A variety of arylboronic acids and amines were converted to the corresponding N-arylazoles and N-arylamines, demonstrating the versatality of the reaction.Keywords
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