Asymmetric Aminohydroxylation of Heteroaromatic Acrylates
- 31 December 1999
- journal article
- letter
- Published by Georg Thieme Verlag KG in Synlett
- Vol. 1999 (12) , 1907-1910
- https://doi.org/10.1055/s-1999-2973
Abstract
N-, S- and O-heteroaromatic acrylates were aminohydroxylated with generally high regio- and enantioselectivity. While pyridylacrylates are not amenable towards this process, the corresponding N-oxides proved to be a useful substitute, allowing the access to biologically important pyridine substituted taxolTM side chain analogs.Keywords
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