Synthesis of potent and selective inhibitors of human plasma kallikrein
- 1 February 1999
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 9 (3) , 301-306
- https://doi.org/10.1016/s0960-894x(98)00562-9
Abstract
No abstract availableKeywords
This publication has 17 references indexed in Scilit:
- On the size of the active site in proteases. I. PapainPublished by Elsevier ,2005
- Synthesis of peptidyl fluoromethyl ketones and peptidyl .alpha.-keto esters as inhibitors of porcine pancreatic elastase, human neutrophil elastase, and rat and human neutrophil cathepsin GJournal of Medicinal Chemistry, 1990
- Synthetic methods and reactions. 141. Fluoride-induced trifluoromethylation of carbonyl compounds with trifluoromethyltrimethylsilane (TMS-CF3). A trifluoromethide equivalentJournal of the American Chemical Society, 1989
- Total synthesis of (.+-.)-15-deoxyspergualinThe Journal of Organic Chemistry, 1987
- Mechanism of slow-binding inhibition of human leukocyte elastase by trifluoromethyl ketonesBiochemistry, 1987
- Reversible, slow, tight-binding inhibition of human Leukocyte elastaseBiochemical and Biophysical Research Communications, 1987
- Fluoro ketone inhibitors of hydrolytic enzymesBiochemistry, 1985
- Refined 2.5 Å X-ray crystal structure of the complex formed by porcine kallikrein A and the bovine pancreatic trypsin inhibitorJournal of Molecular Biology, 1983
- Refined 2 Å X-ray crystal structure of porcine pancreatic kallikrein A, a specific trypsin-like serine proteinaseJournal of Molecular Biology, 1983
- TRANSITION STATE ANALOG INHIBITORS AND ENZYME CATALYSISAnnual Review of Biophysics and Bioengineering, 1976