The erythromycin derivative EM-523 is a potent motilin agonist in man and in rabbit

This publication has 11 references indexed in Scilit:

• Structure‐Activity Relation of Erythromycin‐Related Macrolides in Inducing Contractions and in Displacing Bound Motilin in Rabbit Duodenum
  Neurogastroenterology & Motility, 1989
• Motilides, macrolides with gastrointestinal motor stimulating activity. II. Quaternary N-substituted derivatives of 8,9-anhydroerythromycin A 6,9-hemiacetal and 9,9-dihydroerythromycin A 6,9-epoxide.
  CHEMICAL & PHARMACEUTICAL BULLETIN, 1989
• Motilides, macrolides with gastrointestinal motor stimulating activity. I. O-substituted and tertiary N-substituted derivatives of 8,9-anhydroerythromycin A 6,9-hemiacetal.
  CHEMICAL & PHARMACEUTICAL BULLETIN, 1989
• Comparison of motilin binding to crude homogenates of human and canine gastrointestinal smooth muscle tissue
  Regulatory Peptides, 1988
• Erythromycin and its derivatives with motilin-like biological activities inhibit the specific binding of 125I-motilin to duodenal muscle
  Biochemical and Biophysical Research Communications, 1988
• Macrolides with gastrointestinal motor stimulating activity
  Journal of Medicinal Chemistry, 1987
• Motilin receptors in rabbit stomach and small intestine
  Regulatory Peptides, 1986
• Erythromycin mimics exogenous motilin in gastrointestinal contractile activity in the dog
  American Journal of Physiology-Gastrointestinal and Liver Physiology, 1984
• A simple method for the determination of affinity and binding site concentration in receptor binding studies
  Biochimica et Biophysica Acta (BBA) - Biomembranes, 1977
• Motilin, a Gastric Motor Activity Stimulating Polypeptide: The Complete Amino Acid Sequence
  Canadian Journal of Biochemistry, 1973