Studies on pyrrolidinones. Synthesis of N‐acylpyroglutamic esters with bactericide and fungicide properties
- 1 January 1988
- journal article
- research article
- Published by Wiley in Journal of Heterocyclic Chemistry
- Vol. 25 (1) , 49-57
- https://doi.org/10.1002/jhet.5570250108
Abstract
The best method to prepare N‐acylpyroglutamic esters is to react N‐trimethylsilylpyroglutamic esters with acid chlorides or diketene. These acylesters possess bactericide and fungicide properties against several microorganisms.Keywords
This publication has 41 references indexed in Scilit:
- Chemical conversion of cyclic .ALPHA.-amino acids to .ALPHA.-aminodicarboxylic acids by improved ruthenium tetroxide oxidation.CHEMICAL & PHARMACEUTICAL BULLETIN, 1985
- Synthesis of the Streptomyces ambofaciens antineoplastic constituent 6-diazo-5-oxo-L-norleucineThe Journal of Organic Chemistry, 1983
- SurfactantsAnalytical Chemistry, 1981
- Potent orally active inhibitors of angiotensin-converting enzyme (ACE).CHEMICAL & PHARMACEUTICAL BULLETIN, 1981
- Studies on organometallic compounds. I. Insertion reaction of diketene into N-Si bond of silylated amides.CHEMICAL & PHARMACEUTICAL BULLETIN, 1976
- Syntheses of dl-N-Delnethylvariotinyl 2-Pyrrolidonide (dl-Demethylvariotin), 2-Piperidonide, and ε-CaprolactamideAgricultural and Biological Chemistry, 1973
- Reductive Cyclization of Butyl Pyroglutamate. Synthesis of a New Nitrogen Heterocycle, Decahydrodipyrrolo [a,d]pyrazineJournal of the American Chemical Society, 1952
- Intramolecular Reaction of Acid Chloride and Tertiary Amine GroupsJournal of the American Chemical Society, 1949
- The Hydrogenation of Esters to Alcohols at 25-150°Journal of the American Chemical Society, 1948
- Acetoacetyl ChlorideJournal of the American Chemical Society, 1940