Glycolamide Esters as Biolabile Prodrugs of Carboxylic Acid Agents: Synthesis, Stability, Bioconversion, and Physicochemical Properties
- 1 April 1988
- journal article
- research article
- Published by Elsevier in Journal of Pharmaceutical Sciences
- Vol. 77 (4) , 285-298
- https://doi.org/10.1002/jps.2600770402
Abstract
No abstract availableKeywords
This publication has 54 references indexed in Scilit:
- Esters of N,N-disubstituted 2-hydroxyacetamides as a novel highly biolabile prodrug type for carboxylic acid agentsJournal of Medicinal Chemistry, 1987
- EnalaprilDrugs, 1986
- Enalapril (MK421) activation in man: importance of liver status.Published by Wiley ,1985
- Synthetic and Fermentation-Derived Angiotensin-Converting Enzyme InhibitorsAnnual Review of Pharmacology and Toxicology, 1985
- Clinical Significance of Esterases in ManClinical Pharmacokinetics, 1985
- Esterases: Problems of identification and classificationBiochemical Pharmacology, 1983
- Fenbufen, a New Anti-Inflammatory Analgesic: Synthesis and Structure-Activity Relationships of AnalogsJournal of Pharmaceutical Sciences, 1977
- Rationale for Design of Biologically Reversible Drug Derivatives: ProdrugsJournal of Pharmaceutical Sciences, 1975
- Nonsteroidal antiinflammatory agents. I. 6-Substituted 2-naphthylacetic acidsJournal of Medicinal Chemistry, 1970
- Carboxy Derivatives of Benzylpenicillin1Journal of the American Chemical Society, 1950