Activation of Inhibitors by Sortase Triggers Irreversible Modification of the Active Site
Open Access
- 1 August 2007
- journal article
- Published by Elsevier in Journal of Biological Chemistry
- Vol. 282 (32) , 23129-23139
- https://doi.org/10.1074/jbc.m701857200
Abstract
No abstract availableKeywords
This publication has 56 references indexed in Scilit:
- Rhenium-Catalyzed 1,3-Isomerization of Allylic Alcohols: Scope and Chirality TransferThe Journal of Organic Chemistry, 2006
- Improving the hit-to-lead process: data-driven assessment of drug-like and lead-like screening hitsDrug Discovery Today, 2006
- Synthesis of (2R,3S) 3-amino-4-mercapto-2-butanol, a threonine analogue for covalent inhibition of sortasesBioorganic & Medicinal Chemistry Letters, 2005
- ARP⧸wARP and Automatic Interpretation of Protein Electron Density MapsPublished by Elsevier ,2003
- Irreversible inhibition of the bacterial cysteine protease-transpeptidase sortase (SrtA) by substrate-derived affinity labelsBiochemical Journal, 2002
- A Stereospecific Ruthenium-Catalyzed Allylic AlkylationAngewandte Chemie, 2002
- A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening AssaysSLAS Discovery, 1999
- Palladium-Catalyzed Carbonylative Coupling of Iodonium Salts with Organostannanes under Aqueous Conditions: Synthesis of Unsymmetrical Vinyl and Aromatic KetonesSynthesis, 1998
- Kinetics of the Decomposition of a Mannich BaseJournal of Pharmaceutical Sciences, 1970
- Reactivity of Mannich bases. Part X. The mechanism of the reaction between β-amino-ketones and thiophenolsJournal of the Chemical Society C: Organic, 1967