[3H]OSIP339391, a selective, novel, and high affinity antagonist radioligand for adenosine A2B receptors

This publication has 11 references indexed in Scilit:

• [3H]MRS 1754, a selective antagonist radioligand for A2B adenosine receptors
  Biochemical Pharmacology, 2001
• Why Are A_2BReceptors Low-Affinity Adenosine Receptors? Mutation of Asn273 to Tyr Increases Affinity of Human A_2BReceptor for 2-(1-Hexynyl)adenosine
  Molecular Pharmacology, 2000
• Selective A1-adenosine receptor antagonists identified using yeast Saccharomyces cerevisiae functional assays
  Bioorganic & Medicinal Chemistry Letters, 1999
• An endogenous A_2B adenosine receptor coupled to cyclic AMP generation in human embryonic kidney (HEK 293) cells
  British Journal of Pharmacology, 1997
• Characterization of a 5‐HT_1B receptor on CHO cells: functional responses in the absence of radioligand binding
  British Journal of Pharmacology, 1996
• Monoamine re‐uptake inhibiting 1‐[2‐[(phenoxyphenyl)methoxy]ethyl]‐ piperazines as potential antidepressants
  Recueil des Travaux Chimiques des Pays-Bas, 1993
• Molecular cloning and expression of an adenosine A2b receptor from human brain
  Biochemical and Biophysical Research Communications, 1992
• Identification of Receptors Using Direct Radioligand Binding Techniques
  Published by Springer Nature ,1986
• Quantitative analysis of drug-receptor interactions: I. Determination of kinetic and equilibrium properties
  Life Sciences, 1981
• Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction
  Biochemical Pharmacology, 1973