An efficient synthesis of chlorinated imidazoles throughtert‐butyldimethylsilyloxy derivatives
- 1 September 1994
- journal article
- research article
- Published by Wiley in Journal of Heterocyclic Chemistry
- Vol. 31 (5) , 1121-1123
- https://doi.org/10.1002/jhet.5570310503
Abstract
The protection of 2‐substituted imidazole‐5‐methanol derivatives bytert‐BDMS allowed the chlorination of the heterocycle in position 4 with good yield whereas direct chlorination on the imidazole alcohol was unsuccessful.Keywords
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