Studies of the biogenic amine transporters. II. A brief study on the use of [3H]DA-uptake-inhibition to transporter-binding-inhibition ratios for the in vitro evaluation of putative cocaine antagonists
- 1 January 1993
- journal article
- research article
- Published by Elsevier in Life Sciences
- Vol. 53 (17) , PL267-PL272
- https://doi.org/10.1016/0024-3205(93)90602-y
Abstract
No abstract availableKeywords
This publication has 10 references indexed in Scilit:
- Studies of the biogenic amine transporters. 1. Dopamine reuptake blockers inhibit [3H]mazindol binding to the dopamine transporter by a competitive mechanism: Preliminary evidence for different binding domainsNeurochemical Research, 1994
- Identification of a GBR12935 homolog, LR1111, which is over 4,000‐fold selective for the dopamine transporter, relative to serotonin and norepinephrine transportersSynapse, 1993
- Cocaine and GBR12909 produce equivalent motoric responses at different occupancy of the dopamine transporterPharmacology Biochemistry and Behavior, 1992
- GBR12909 antagonizes the ability of cocaine to elevate extracellular levels of dopaminePharmacology Biochemistry and Behavior, 1991
- Synthesis, ligand binding, QSAR, and CoMFA study of 3.beta.-(p-substituted phenyl)tropane-2.beta.-carboxylic acid methyl estersJournal of Medicinal Chemistry, 1991
- The dopamine hypothesis of the reinforcing properties of cocaineTrends in Neurosciences, 1991
- [125I]RTI-55: a potent ligand for dopamine transportersEuropean Journal of Pharmacology, 1991
- [3H]GBR 12935 binding in vivo in mouse brain: labelling of a piperazine acceptor siteEuropean Journal of Pharmacology, 1987
- Cocaine Receptors on Dopamine Transporters Are Related to Self-Administration of CocaineScience, 1987
- PROTEIN MEASUREMENT WITH THE FOLIN PHENOL REAGENTJournal of Biological Chemistry, 1951