Synthesis of analogs of the carboxyl protease inhibitor pepstatin. Effect of structure on inhibition of pepsin and renin
- 1 January 1980
- journal article
- research article
- Published by American Chemical Society (ACS) in Journal of Medicinal Chemistry
- Vol. 23 (1) , 27-33
- https://doi.org/10.1021/jm00175a006
Abstract
Note: In lieu of an abstract, this is the article's first page.This publication has 8 references indexed in Scilit:
- Synthesis of all the stereoisomers of statine (4-amino-3-hydroxy-6-methylheptanoic acid). Inhibition of pepsin activity by N-carbobenzoxy-L-valyl-L-valyl-statine derived from the four stereoisomersJournal of Medicinal Chemistry, 1979
- Pepsin inhibition by a high specific activity radioiodinated derivative of pepstatinArchives of Biochemistry and Biophysics, 1979
- Synthesis of (3S,4S)-4-amino-3-hydroxy-6-methylheptanoic acid derivatives. Analysis of diastereomeric purityThe Journal of Organic Chemistry, 1978
- Synthesis of dideoxy-pepstatin. Mechanism of inhibition of porcine pepsinBiochemical and Biophysical Research Communications, 1977
- Mode of inhibition of acid proteases by pepstatin.Journal of Biological Chemistry, 1976
- The crystal structure at 5.5Å resolution of an acid-protease from Rhizopus chinensisBiochemical and Biophysical Research Communications, 1976
- N-Acylated derivatives of a peptide obtained by enzymatic degradation of pepstatins.The Journal of Antibiotics, 1975
- Un substrat pour le dosage chimique de la rénineHelvetica Chimica Acta, 1966