New sialyltransferase inhibitors based on CMP-quinic acid: development of a new sialyltransferase assay
- 1 January 1998
- journal article
- Published by Springer Nature in Glycoconjugate Journal
- Vol. 15 (4) , 345-354
- https://doi.org/10.1023/a:1006917717161
Abstract
Quinic acid (4) was transformed into phosphitamides 6, 14, and 15, which could be readily linked to 5′-O-unprotected cytidine derivative 7; ensuing oxidation of the obtained phosphite triesters with...Keywords
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