Synthesis and evaluation of [18F] labeled benzamides: High affinity sigma receptor ligands for PET imaging

This publication has 17 references indexed in Scilit:

• Sigma receptors are expressed in human non-small cell lung carcinoma
  Life Sciences, 1995
• Regional variation in the ratio of σ1 to σ2 binding in rat brain
  European Journal of Pharmacology, 1994
• Rat liver and kidney contain high densities of σ1 and σ2 receptors: characterization by ligand binding and photoaffinity labeling
  European Journal of Pharmacology: Molecular Pharmacology, 1994
• Synthesis and Characterization of [125I]-N-(N-Benzylpiperidin-4-yl)-4-iodobenzamide, a New .sigma. Receptor Radiopharmaceutical: High-Affinity Binding to MCF-7 Breast Tumor Cells
  Journal of Medicinal Chemistry, 1994
• The use of [18F]4-fluorobenzyl iodide (FBI) in PET radiotracer synthesis: Model alkylation studies and its application in the design of dopamine D1 and D2 receptor-based imaging agents
  Nuclear Medicine and Biology, 1993
• An improved synthesis of [125I]N-(diethylaminoethyl)-4-iodobenzamide: a potential ligand for imaging malignant melanoma
  Nuclear Medicine and Biology, 1993
• A sigma-like binding site in rat pheochromocytoma (PC12) cells: decreased affinity for (+)-benzomorphans and lower molecular weight suggest a different sigma receptor form from that of guinea pig brain
  Brain Research, 1990
• Autoradiographic visualization of haloperidol-sensitive sigma receptors in guinea-pig brain
  Neuroscience, 1988
• Autoradiographic localization of sigma receptor binding sites in guinea pig and rat central nervous system with (+)3H-3-(3-hydroxyphenyl)-N-(1- propyl)piperidine
  Journal of Neuroscience, 1986
• An improved [18O]water target for[[18F]fluoride production
  The International Journal of Applied Radiation and Isotopes, 1985