Synthesis of Phosphonic Acid Analogues of Sialic Acids (Neu5Ac and KDN) as Potential Sialidase Inhibitors
- 1 May 1997
- journal article
- Published by American Chemical Society (ACS) in The Journal of Organic Chemistry
- Vol. 62 (11) , 3500-3504
- https://doi.org/10.1021/jo961891p
Abstract
No abstract availableKeywords
This publication has 14 references indexed in Scilit:
- Design and Synthesis of Sialyl Lewis X MimeticsJournal of the American Chemical Society, 1995
- The first synthesis of a C-7 nitrogen-containing sialic acid analogue,
acetamido-7-azido-3,5,7-trideoxy- -glycero-d d nonulopyranosonic acid (7-azido-7-deoxy-Neu5Ac)Tetrahedron Letters, 1995 - Crystal structure of Vibrio cholerae neuraminidase reveals dual lectin-like domains in addition to the catalytic domainStructure, 1994
- Molecular Modeling Studies on Ligand Binding to Sialidase from Influenza Virus and the Mechanism of CatalysisJournal of Medicinal Chemistry, 1994
- Indium-mediated allylations of unprotected carbohydrates in aqueous media: a short synthesis of sialic acidThe Journal of Organic Chemistry, 1993
- Rational design of potent sialidase-based inhibitors of influenza virus replicationNature, 1993
- Chemical-enzymic synthesis and conformational analysis of sialyl Lewis X and derivativesJournal of the American Chemical Society, 1992
- A concise chemical synthesis of (+)-3-deoxy-D-glycero-D-galacto-nonulosonic acid (KDN)Journal of the Chemical Society, Chemical Communications, 1992
- Synthesis of a Phosphonic Acid Analogue of N‐Acetyl‐2,3‐didehydro‐2‐deoxyneuraminic Acid, an Inhibitor of Vibrio cholerae SialidaseHelvetica Chimica Acta, 1991
- Addition of functionalized allylic bromides to terminal alkynesTetrahedron Letters, 1984