Regioselective synthesis of a-ring halogenated derivatives of 17α-ethynyloestradiol

This publication has 21 references indexed in Scilit:

• Efficient regioselective a-ring functionalization of oestrogens
  Tetrahedron, 1990
• 2-bromo- and 16-bromo-estrogens and related compounds: Potential inhibitors for both estradiol 2- and 16α-hydroxylases in rat liver microsomes
  The Journal of Steroid Biochemistry and Molecular Biology, 1989
• Drug protein conjugates—III. Inhibition of the irreversible binding of ethinylestradiol to rat liver microsomal protein by mixed-function oxidase inhibitors, ascorbic acid and thiols
  The Journal of Steroid Biochemistry and Molecular Biology, 1983
• Drug-protein conjugates—V
  Biochemical Pharmacology, 1983
• The biliary and urinary metabolites of [3H]17α-ethynylestradiol in women
  Xenobiotica, 1983
• The biotransformation of 17α-ethynyl[³H]estradiol in the rat: Irreversible binding and biliary metabolites
  Xenobiotica, 1982
• Comparative Study of Ethynyloestradiol Metabolism in the Rabbit, Guinea Pig and Rat
  Hormone Research, 1979
• Metabolism of 17α-Ethinylestradiol by Human Liver Microsomesin Vitro: Aromatic Hydroxylation and Irreversible Protein Binding of Metabolites
  Journal of Clinical Endocrinology & Metabolism, 1974
• Studies on the Metabolism of Ethynylestradiolin vitroandin vivo: The Significance of 2-Hydroxylation and the Formation of Polar Products
  Xenobiotica, 1973
• 2,4-Dibromo-α-oestradiol
  Journal of the American Chemical Society, 1940