1-(Phenylsulfonyl)indol-2-yl Triflate: A Versatile Reagent for the Synthesis of 2-Substituted Indoles
- 1 September 1996
- journal article
- research article
- Published by Taylor & Francis in Synthetic Communications
- Vol. 26 (17) , 3289-3295
- https://doi.org/10.1080/00397919608004639
Abstract
The palladium-catalysed reaction of 1-(phenylsulfonyl)indol-2-yl triflate 1, with a variety of aryl and heteroaryl boronic acids 2 or vinyl tributylstannane 3 provides a general and an efficient method for the synthesis of 2-substituted indoles 4.Keywords
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