A mild and convenient method for tritium labelling of activated aromatic compounds using BF3–Et2O and tritiated water
- 1 January 1993
- journal article
- research article
- Published by Royal Society of Chemistry (RSC) in Journal of the Chemical Society, Chemical Communications
- No. 9,p. 774-776
- https://doi.org/10.1039/c39930000774
Abstract
A procedure for tritium exchange labelling of activated aromatic compounds using 3H2O and BF3–Et2O has been developed to prepare two radio-labelled photoprobes that are difficult to obtain by conventional methods; the applicability of the method has been examined by labelling several aromatic compounds varying in activation toward electrophilic aromatic substitution.Keywords
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