GR159897 and related analogues as highly potent, orally active non-peptide neurokinin NK2 receptor antagonists.
- 25 August 1994
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 4 (16) , 1951-1956
- https://doi.org/10.1016/s0960-894x(01)80541-2
Abstract
No abstract availableKeywords
This publication has 11 references indexed in Scilit:
- Characterisation, CNS distribution and function of NK2 receptors studied using potent NK2 receptor antagonistsRegulatory Peptides, 1993
- Low molecular weight neurokinin NK2 antagonistsBioorganic & Medicinal Chemistry Letters, 1993
- A potent and selective non-peptide antagonist of the neurokinin a (NK2) receptorLife Sciences, 1992
- Conformationally constrained tachykinin analogs: potent and highly selective neurokinin NK-2 receptor agonistsJournal of Medicinal Chemistry, 1992
- Highly potent and selective heptapeptide antagonists of the neurokinin NK-2 receptorJournal of Medicinal Chemistry, 1992
- A general route to enantiomerically pure sulfoxides from a chiral sulfiteThe Journal of Organic Chemistry, 1991
- Total syntheses of yohimbe alkaloids, with stereoselection for the normal, allo, and 3-epiallo series, based on annelations of 4-methoxy-1,2-dihydropyridonesThe Journal of Organic Chemistry, 1991
- Chapter 5. Recent Advances in Neurokinin Receptor AntagonistsPublished by Elsevier ,1991
- TachykininsAnnual Review of Neuroscience, 1988
- A rapid, simple, and mild procedure for alkylation of phenols, alcohols, amides and acidsTetrahedron, 1979