An Improved Synthesis of Chiral α-(4-Bromobenzyl)alanine Ethyl Ester and Its Application to the Synthesis of LFA-1 Antagonist BIRT-377

This publication has 9 references indexed in Scilit:

• Self-Regeneration of Stereocenters: A Practical Enantiospecific Synthesis of LFA-1 Antagonist BIRT-377
  Organic Letters, 2000
• Self‐Regeneration of Stereocenters (SRS)—Applications, Limitations, and Abandonment of a Synthetic Principle
  Angewandte Chemie International Edition in English, 1996
• A short asymmetric synthesis of N-α-fmoc-N-δ-boc-α-methyl-D-ornithine
  Bioorganic & Medicinal Chemistry Letters, 1995
• Enantiospecific conversion of (S)-alanine to (R)-α-methyl phenylalanine
  Tetrahedron: Asymmetry, 1995
• A Facially-Selective Protonation Controls the Stereochemistry of a Key Intermediate in the Synthesis of 1.beta.-Methylcarbapenems
  The Journal of Organic Chemistry, 1994
• α-Alkylation of acyclic amino acids with self-reproduction of the Center of Chirality. A new route to (S)-(+)-α-alkylated aspartic acids.
  Tetrahedron Letters, 1987
• N,O‐Acetals from Pivalaldehyde and Amino Acids for the α‐Alkylation with Self‐Reproduction of the Center of Chirality. Enolates of 3‐Benzoyl‐2‐(tert‐butyl)‐1,3‐oxazolidin‐5‐ones
  Helvetica Chimica Acta, 1985
• Enantioretentive alkylation of acyclic amino acids
  Tetrahedron Letters, 1984
• Peptidsynthesen nach dem Oxazolidon‐Verfahren, III
  European Journal of Inorganic Chemistry, 1959