Incorporation of a phosphonic acid isostere of aspartic acid into peptides using Fmoc-solid phase synthesis
- 9 April 1998
- journal article
- Published by Elsevier in Tetrahedron Letters
- Vol. 39 (15) , 2067-2070
- https://doi.org/10.1016/s0040-4039(98)00189-0
Abstract
No abstract availableKeywords
This publication has 18 references indexed in Scilit:
- Solid phase synthesis of peptides containing the non-hydrolysable analog of (O)phosphotyrosine, P(CH2PO3H2)PheInternational Journal of Peptide and Protein Research, 2009
- Farnesyl Diphosphate-Based Inhibitors of Ras Farnesyl Protein TransferaseJournal of Medicinal Chemistry, 1995
- Deprotection and cleavage methods for protected peptide resins containing 4-[(diethylphosphono)difluoromethyl]-D,L-phenylalanine residuesTetrahedron Letters, 1993
- A short synthesis of (S)-3-(dimethylphosphono)-2- ((9-fluorenyl)methoxycarbamoyl)propionic acid, a protected phosphonic acid analogue of aspartic acidTetrahedron Letters, 1992
- Asymmetric Synthesis of (1-Aminoalkyl)phosphonic Acids via Asymmetric Aldol Reaction of (Isocyanomethyl)phosphonates Catalyzed by a Chiral Ferrocenylphosphine-Gold(I) ComplexTetrahedron Letters, 1989
- Methotrexate analog. 32. Chain extension, .alpha.-carboxyl deletion, and .gamma. carboxyl replacement by sulfonate and phosphate. Effect on enzyme binding and cell-growth inhibitionJournal of Medicinal Chemistry, 1988
- An efficient synthesis of γ-amino-β-ketoalkylphosphonates from α-amino acidsTetrahedron Letters, 1987
- N-(Phosphonoacetyl)amino phosphonates. Phosphonate analogs of N-(phosphonoacetyl)-L-aspartic acid (PALA)Journal of Medicinal Chemistry, 1985
- Phosphorous-Containing Analogues of AspartameJournal of Pharmaceutical Sciences, 1984
- Phosphonodipeptides: synthesis and separation of diastereoisomersCanadian Journal of Chemistry, 1982