Iterative Approach to the Discovery of Novel Degarelix Analogues: Substitutions at Positions 3, 7, and 8. Part II
- 28 June 2005
- journal article
- research article
- Published by American Chemical Society (ACS) in Journal of Medicinal Chemistry
- Vol. 48 (15) , 4851-4860
- https://doi.org/10.1021/jm050134t
Abstract
No abstract availableKeywords
This publication has 49 references indexed in Scilit:
- Novel gonadotropin‐releasing hormone antagonists with substitutions at position 5Peptide Science, 2004
- Reductive Amination of Aldehydes and Ketones with Sodium Triacetoxyborohydride. Studies on Direct and Indirect Reductive Amination Procedures1The Journal of Organic Chemistry, 1996
- Design, synthesis and bioassays of antagonists of LHRH which have high antiovulatory activity and release negligible histamineBiochemical and Biophysical Research Communications, 1987
- Effect of reductive alkylation of lysine in positions 6 and/or 8 on the histamine-releasing activity of luteinizing hormone-releasing hormone antagonistsJournal of Medicinal Chemistry, 1987
- Improved antagonists of luteinizing hormone-releasing hormone modified in position 7Journal of Medicinal Chemistry, 1985
- Isolation and characterization of chicken hypothalamic luteinizing hormone-releasing hormoneBiochemical and Biophysical Research Communications, 1982
- Luteinizing hormone-releasing hormone. Antiovulatory activity of analogs substituted in positions 2 and 6Journal of Medicinal Chemistry, 1975
- Analogs of luteinizing hormone releasing factor (LRF) synthesis and biological activity of [(Nα-Me)Leu7]LRF and [D-Ala6,(Nα-Me)Leu7]LRFBiochemical and Biophysical Research Communications, 1975
- 1339. Substituted diphenylmethyl protecting groups in peptide synthesisJournal of the Chemical Society, 1965
- BOOK REVIEWSJournal of the American Chemical Society, 1953