Synthesis, inhibitory activity towards human leukocyte elastase and molecular modelling studies of 1-carbamoyl-4-methyleneaminoxyazetidinones
- 1 January 2000
- journal article
- Published by Elsevier in European Journal of Medicinal Chemistry
- Vol. 35 (1) , 53-67
- https://doi.org/10.1016/s0223-5234(00)00111-2
Abstract
No abstract availableKeywords
This publication has 35 references indexed in Scilit:
- Discovery and Biological Activity of Orally Active Peptidyl Trifluoromethyl Ketone Inhibitors of Human Neutrophil ElastaseJournal of Medicinal Chemistry, 1997
- Peptidyl .alpha.-ketoheterocyclic inhibitors of human neutrophil elastase. 2. Effect of varying the heterocyclic ring on in vitro potencyJournal of Medicinal Chemistry, 1995
- Inhibition of Human Neutrophil Elastase. 3. An Orally Active Enol Acetate ProdrugJournal of Medicinal Chemistry, 1995
- Proteinases in Chronic Lung InfectionaAnnals of the New York Academy of Sciences, 1991
- Neutrophil ProteinasesAnnals of the New York Academy of Sciences, 1991
- Putative Role of Neutrophil Elastase in the Pathogenesis of EmphysemaaAnnals of the New York Academy of Sciences, 1991
- Degradation of connective tissue components by lung derived leucocytes in vitro: role of proteases and oxidants.Thorax, 1988
- Elastase and alpha 1-proteinase inhibitor activity in tracheal aspirates during respiratory distress syndrome. Role of inflammation in the pathogenesis of bronchopulmonary dysplasia.Journal of Clinical Investigation, 1983
- Human neutrophil elastase functions as a type III collagen “Collagenase”Biochemical and Biophysical Research Communications, 1980
- MEDIATORS OF INFLAMMATION IN LEUKOCYTE LYSOSOMESThe Journal of Experimental Medicine, 1968