Inhibitors of the acrosomal proteinase acrosin: Human urinary trypsin inhibitor (UTI) and 4-(2-carboxyethyl) phenyl trans 4-aminomethylcyclohexanecarboxylate hydrochloride (DV-1006)
- 1 September 1980
- journal article
- research article
- Published by Springer Nature in Cellular and Molecular Life Sciences
- Vol. 36 (9) , 1103-1104
- https://doi.org/10.1007/bf01965994
Abstract
Human urinary trypsin inhibitor (UTI) and (4-(2-carboxyethyl) phenyl trans 4-aminoethylcyclohexanecarboxylate hydrochloride (DV-1006) competitively inhibited the human acrosomal proteinase acrosin; Ki values were 1.2×10−8M and 9.4×10−7 M, respectively.This publication has 8 references indexed in Scilit:
- Studies on human urinary trypsin inhibitor 1. Its modification on treatment of urine with acidThrombosis Research, 1977
- [Trypsin inhibitors in human urine (author's transl)].1977
- Proteinase Inhibitors in Human Cervical Mucus and Their in vitro Interactions with Human AcrosinPublished by Springer Nature ,1974
- Proteinase Inhibitors of the Respiratory Tract: Studies on the Structural Relationship between Acid-Stable Inhibitors Present in the Respiratory Tract, Plasma and UrinePublished by Springer Nature ,1974
- Leupeptin and Antipain. Strong Competitive Inhibitors of Sperm Acrosomal Proteinase (Boar Acrosin) and Kallikreins from Porcine Organs (Pancreas, Submand. Glands, Urine)Hoppe-Seyler´s Zeitschrift Für Physiologische Chemie, 1973
- Acrosomal Proteinase and Proteinase Inhibitor of Human SpermatozoaScience, 1972
- Inhibitory effects of ω-amino acid esters on trypsin, plasmin, plasma kallikrein and thrombinBiochimica et Biophysica Acta (BBA) - Enzymology, 1971
- The determination of enzyme inhibitor constantsBiochemical Journal, 1953