Cyclic and acyclic partial retro-inverso enkephalinamides: Mu receptor selective enzyme resistant analogs
- 1 September 1983
- journal article
- research article
- Published by Elsevier in Biochemical and Biophysical Research Communications
- Vol. 115 (3) , 864-870
- https://doi.org/10.1016/s0006-291x(83)80014-x
Abstract
No abstract availableKeywords
This publication has 16 references indexed in Scilit:
- Synthesis and pharmacological characterization in vitro of cyclic enkephalin analogs: effect of conformational constraints on opiate receptor selectivityJournal of Medicinal Chemistry, 1982
- Conformational restrictions of biologically active peptides via amino acid side chain groupsLife Sciences, 1982
- Opiate receptor subclasses differ in their conformational requirementsNature, 1982
- Structure-Activity Relationships of Enkephalin-Like PeptidesAnnual Review of Pharmacology and Toxicology, 1980
- Unsulfated C-terminal 7-peptide of cholecystokinin: A new ligand of the opiate receptorBiochemical and Biophysical Research Communications, 1978
- High-affinity enkephalin-degrading peptidase in brain is increased after morphineNature, 1978
- Endogenous opioid peptides: multiple agonists and receptorsNature, 1977
- [D-Ala 2 ]-Met-Enkephalinamide: A Potent, Long-Lasting Synthetic Pentapeptide AnalgesicScience, 1976
- Identification of two related pentapeptides from the brain with potent opiate agonist activityNature, 1975
- Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reactionBiochemical Pharmacology, 1973