Iterative Amination Strategy in the Synthesis of Peptidomimetics
- 1 November 1997
- journal article
- Published by Oxford University Press (OUP) in Chemistry Letters
- Vol. 26 (11) , 1159-1160
- https://doi.org/10.1246/cl.1997.1159
Abstract
An iterative palladium catalysed cross-coupling reaction of aryl bromides with amines has been employed in the preparation of novel peptidomimetics. This is a versatile strategy with which we can demonstrate the principle of library synthesis by using a diverse range of coupling partnersKeywords
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