Synthesis of 1α, 25-Dihydroxyvitamin D3 A-Ring Synthon by Pd-Catalyzed Cyclization

Abstract
A short and efficient synthesis of 1α, 25-dihydroxyvitamin D3 A-ring synthon starting from diketene, acrolein and ethyl malonate by using palladium-catalyzed cyclization of the (Z)-enol triflate is described.

This publication has 0 references indexed in Scilit: