Studies Directed to the Total Synthesis of ET 743 and Analogues Thereof: An Expeditious Route to the ABFGH Subunit
- 13 December 2001
- journal article
- letter
- Published by American Chemical Society (ACS) in Organic Letters
- Vol. 4 (1) , 43-46
- https://doi.org/10.1021/ol016844k
Abstract
In model studies directed to the total synthesis of Et743, a strategic S−C bond formation in systems 26 and 27 was demonstrated. It was further shown that Pictet−Spengler cyclization leading to spiro product 33 exhibits very high stereoselection.Keywords
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