A Practical Synthesis of Geometrically PureN-Boc-Protected Primary Allylic Amines
- 1 January 1994
- journal article
- letter
- Published by Georg Thieme Verlag KG in Synlett
- Vol. 1994 (05) , 368-370
- https://doi.org/10.1055/s-1994-22857
Abstract
N-Boc-Protected primary allylic amines are easily prepared from the corresponding mesylates or halides by using di-tert-butyl imidodicarbonate (Boc2NH) and K2CO3 or Cs2CO3 in a Gabriel-type substitution, followed by selective removal of one Boc group with TFA.Keywords
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