Synthesis of (1α,5α,6α)-6-Amino-3-azabicyclo[3.1.0]hexane, a Novel Achiral Diamine

Abstract
Synthesis of (1α,5α,6α)-6-amino-3-azabicyclo[3.1.0]hexane is described. Ethyl diazoacetate cycloaddition to a pyrroline or maleimide derivative provides the azabicyclohexyl system; amine introduction is then effected using a modified Curtius rearrangement.

This publication has 0 references indexed in Scilit: