Preparation of N-protected α-amino alcohols by acetoxyborohydride reduction of N-protected α-amino acid esters

Abstract
N-Protected α-amino alcohols were prepared by reduction of N-protected α-amino acid esters by sodium acetoxyborohydride in dioxane at elevated temperature. The reductions proceed with excellent yields and without racemisation. Reduction of the carbamate protecting groups was not observed.

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