SOME IN VITRO INHIBITORS OF CARBONIC ANHYDRASE
- 1 September 1958
- journal article
- Published by Oxford University Press (OUP) in Journal of Pharmacy and Pharmacology
- Vol. 10 (1) , 696-705
- https://doi.org/10.1111/j.2042-7158.1958.tb10362.x
Abstract
Work on sulphonamides as in vitro inhibitors of carbonic anhydrase has been extended by the preparation and assay of novel types. Although diphenylsulphonamides, p-alkoxycarbonylbenzene sulphonamides and 5-alkoxycarbonylamino-1:3:4-thiadiazole-2-sulphon-amides showed noteworthy activity in vitro, only the thiadiazole derivatives possessed diuretic activity in the rat.Keywords
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