Sialidase inhibitors related to zanamivir. Further SAR studies of 4-amino-4H-pyran-2-carboxylic acid-6-propylamides
- 8 March 2001
- journal article
- research article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 11 (5) , 669-673
- https://doi.org/10.1016/s0960-894x(01)00019-1
Abstract
No abstract availableKeywords
This publication has 14 references indexed in Scilit:
- In-vitro and in-vivo efficacy of influenza neuraminidase inhibitorsCurrent Opinion in Infectious Diseases, 1998
- Structure−Activity Relationship Studies of Novel Carbocyclic Influenza Neuraminidase InhibitorsJournal of Medicinal Chemistry, 1998
- Dihydropyrancarboxamides Related to Zanamivir: A New Series of Inhibitors of Influenza Virus Sialidases. 2. Crystallographic and Molecular Modeling Study of Complexes of 4-Amino-4H-pyran-6-carboxamides and Sialidase from Influenza Virus Types A and BJournal of Medicinal Chemistry, 1998
- Dihydropyrancarboxamides Related to Zanamivir: A New Series of Inhibitors of Influenza Virus Sialidases. 1. Discovery, Synthesis, Biological Activity, and Structure−Activity Relationships of 4-Guanidino- and 4-Amino-4H-pyran-6-carboxamidesJournal of Medicinal Chemistry, 1998
- ZanamivirDrugs, 1998
- A regio- and stereo-selective introduction of azide at C-4 of 2,3-unsaturated N-acetylneuraminic acidsCarbohydrate Research, 1997
- Influenza Neuraminidase Inhibitors Possessing a Novel Hydrophobic Interaction in the Enzyme Active Site: Design, Synthesis, and Structural Analysis of Carbocyclic Sialic Acid Analogues with Potent Anti-Influenza ActivityJournal of the American Chemical Society, 1997
- Structural Variations on N‐acetylneuraminic acid, 20. Synthesis of some 2,3‐didehydro‐2‐deoxysialic Acids structurally varied at C‐4 and their behavior towards Sialidase from Vibrio choleraeEuropean Journal of Organic Chemistry, 1991
- New coupling reagents in peptide chemistryTetrahedron Letters, 1989
- A Stereospecific Synthesis of β-Glycosides of N-Acetylneuraminic Acid and Secondary AlcoholsChemistry Letters, 1986