The kappa-active oxygen in the opioid pharmacophore of some benzomorphans: Charges, proton affinties and binding modelling
- 1 December 1984
- journal article
- research article
- Published by Elsevier in Neuropeptides
- Vol. 5 (1-3) , 209-212
- https://doi.org/10.1016/0143-4179(84)90064-7
Abstract
No abstract availableKeywords
This publication has 4 references indexed in Scilit:
- 5-Ethyl-2'-hydroxy-2-[(1-hydroxycyclopropyl)methyl]-9,9-dimethyl-6,7-benzomorphan hydrochloride (bremazocine), C20H29NO2.HClActa Crystallographica Section C Crystal Structure Communications, 1984
- Structural studies of substituted 6,7-benzomorphan compounds. VI. (−)-(1R,5R,9R,13R)-2'-Hydroxy-5,9α-dimethyl-2-(tetrahydrofurfuryl)-6,7-benzomorphan and (−)-(1R,5R,9R,13S)-2'-hydroxy-5,9-dimethyl-2-(tetrahydrofurfuryl)-6,7-benzomorphan tartrate monohydrateActa Crystallographica Section B: Structural Science, Crystal Engineering and Materials, 1982
- N-[(Tetrahydrofuryl)alkyl] and N-(alkoxyalkyl) derivatives of (-)-normetazocine, compounds with differentiated opioid action profilesJournal of Medicinal Chemistry, 1979
- Quantum chemical studies of morphine-like opiate narcotics. Effect of N-substituent variationsJournal of Medicinal Chemistry, 1975