Use of Metabolite AUC Data in Bioavailability Studies to Discriminate Between Absorption and First-Pass Extraction
- 1 May 1990
- journal article
- Published by Springer Nature in Clinical Pharmacokinetics
- Vol. 18 (5) , 419-422
- https://doi.org/10.2165/00003088-199018050-00006
Abstract
No abstract availableKeywords
This publication has 11 references indexed in Scilit:
- A general model of metabolite kinetics following intravenous and oral administration of the parent drugBiopharmaceutics & Drug Disposition, 1988
- Pharmacokinetics of Diphenhydramine and a Demethylated Metabolite Following Intravenous And Oral AdministrationThe Journal of Clinical Pharmacology, 1986
- Metabolite residence time: influence of the first-pass effect.1986
- Pharmacokinetics of ketanserin and its metabolite ketanserin-ol in man after intravenous, intramuscular and oral administrationEuropean Journal of Clinical Pharmacology, 1986
- Disposition of nomifensine after acute and prolonged dosingClinical Pharmacology & Therapeutics, 1986
- Influence of dose and route of administration on disposition of metronidazole and its major metabolitesEuropean Journal of Clinical Pharmacology, 1986
- A review of metabolite kineticsJournal of Pharmacokinetics and Biopharmaceutics, 1985
- Pharmacokinetics of triamterene after i.v. administration to man: Determination of bioavailabilityEuropean Journal of Clinical Pharmacology, 1983
- Studies of the different metabolic pathways of antipyrine in manEuropean Journal of Clinical Pharmacology, 1982
- Pharmacokinetics of lidocaine and its deethylated metabolite: Dose and time dependency studies in manJournal of Pharmacokinetics and Biopharmaceutics, 1982