First Report of the Investigation into the Importance of pKa in the Inhibition of Estrone Sulfatase by Sulfamate Containing Compounds
- 7 June 2000
- journal article
- Published by Elsevier in Biochemical and Biophysical Research Communications
- Vol. 272 (2) , 583-585
- https://doi.org/10.1006/bbrc.2000.2812
Abstract
No abstract availableKeywords
This publication has 8 references indexed in Scilit:
- Steroidal and Nonsteroidal Sulfamates as Potent Inhibitors of Steroid SulfataseJournal of Medicinal Chemistry, 1998
- Steroid sulphatase: expression, isolation and inhibition for active-site identification studiesChemico-Biological Interactions, 1998
- Estrone sulfonates as inhibitors of estrone sulfataseSteroids, 1997
- Estrone Sulfatase: Probing Structural Requirements for Substrate and Inhibitor RecognitionBiochemistry, 1997
- Inhibition of placental estrone sulfatase activity and MCF-7 breast cancer cell proliferation by estrone-3-amino derivativesThe Journal of Steroid Biochemistry and Molecular Biology, 1996
- Heteroatom-substituted analogues of the active-site directed inhibitor estra-1,3,5(10)-trien-17-one-3-sulphamate inhibit estrone sulphatase by a different mechanismThe Journal of Steroid Biochemistry and Molecular Biology, 1996
- Estrone sulfate analogs as estrone sulfatase inhibitorsSteroids, 1995
- Aromatase inhibitors and their potential clinical significanceJournal of Steroid Biochemistry, 1986